Suprastin analogues of the drug

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Suprastin - instructions for use, analogs, reviews and release forms (25 mg tablets, injections) medications for the treatment of urticaria, itching and other allergic diseases in adults, children (including newborns) and during pregnancy

In this article you can read the instructions for use of the drug Suprastin.

Table of contents:

Reviews of site visitors - consumers of this medicine, as well as the opinions of specialist doctors on the use of Suprastin in their practice are presented. We kindly ask you to actively add your reviews about the drug: whether the medicine helped or did not help get rid of the disease, what complications and side effects were observed, perhaps not stated by the manufacturer in the annotation. Suprastin analogues in the presence of existing structural analogues. Use for the treatment of urticaria, dermatitis, allergies, itching and other allergic diseases and conditions in adults, children (including newborns), as well as during pregnancy and lactation.

Suprastin is a histamine H1 receptor blocker, an ethylenediamine derivative. Prevents the development and facilitates the course of allergic reactions. It has a moderate sedative and pronounced antipruritic effect. It has an antiemetic effect, peripheral anticholinergic activity, and moderate antispasmodic properties.

The therapeutic effect develops within minutes after oral administration, reaches a maximum within the first hour after administration and lasts at least 3-6 hours.

After oral administration, chloropyramine hydrochloride is quickly and completely absorbed from the gastrointestinal tract. Intensively metabolized in the liver. It is excreted primarily in the urine in the form of metabolites.

In children, drug elimination occurs faster than in adults.

  • hives;
  • angioedema (Quincke's edema);
  • serum sickness;
  • seasonal and year-round allergic rhinitis;
  • conjunctivitis;
  • contact dermatitis;
  • skin itching;
  • acute and chronic eczema;
  • atopic dermatitis;
  • food and drug allergies;
  • allergic reactions to insect bites.

Solution for intramuscular and intravenous injections (injections) 20 mg/ml.

Instructions for use and dosage

Orally, during meals, without chewing and with plenty of water.

Adults: prescribe 1 tablet. 3-4 times a day (mg/day).

Children: aged 1 to 12 months - 1/4 tablet. (6.5 mg) 2-3 times a day (ground to powder form along with baby food); from 1 to 6 years - 1/4 of the table. 3 times a day or 1/2 tablet. 2 times a day; from 6 to 14 years - 1/2 table. (12.5 mg) 2-3 times a day.

The dose can be gradually increased if the patient has no side effects, but the maximum dose should never exceed 2 mg/kg body weight.

Injection:

IM, IV (used only in acute severe cases under the supervision of a physician!)

Adults: recommended daily dose (1-2 amps) IM.

Children aged 1 to 12 months: recommended initial doses - 0.25 ml (1/4 ampoule) IM; from 1 to 6 years - 0.5 ml (1/2 amp) IM; from 6 to 14 years - 0.5-1 ml (1/2-1 amp.) IM.

The dose may be increased cautiously depending on the patient's response and observed side effects. However, the dose should never exceed 2 mg/kg. In case of severe allergies, treatment should begin with a careful, slow intravenous injection, and then continue with intramuscular injections or oral administration of the drug.

Special groups of patients (general recommendations for both forms)

Elderly, debilitated patients: the use of the drug Suprastin requires special caution, because in these patients, antihistamines are more likely to cause side effects (dizziness, drowsiness).

Patients with impaired liver function: a dose reduction may be required due to a decrease in the metabolism of the active component of the drug in liver diseases.

Patients with impaired renal function: a change in the dosage regimen and a dose reduction may be required due to the fact that the active component is mainly excreted through the kidneys.

  • drowsiness;
  • fatigue;
  • dizziness;
  • nervous excitement;
  • tremor;
  • headache;
  • euphoria;
  • abdominal discomfort;
  • dry mouth;
  • nausea, vomiting;
  • diarrhea, constipation;
  • loss or increase in appetite;
  • decrease in blood pressure;
  • tachycardia;
  • leukopenia, agranulocytosis;
  • muscle weakness;
  • increased intraocular pressure;
  • photosensitivity.

Side effects occur, as a rule, extremely rarely, are temporary and disappear after discontinuation of the drug.

  • acute attack of bronchial asthma;
  • pregnancy;
  • lactation (breastfeeding);
  • newborns (including premature babies);
  • hypersensitivity to the drug or other ethylenediamine derivatives.

Use during pregnancy and breastfeeding

There have been no adequate and well-controlled studies of the use of antihistamines during pregnancy. Therefore, the use of the drug in pregnant women (especially in the 1st trimester and the last month of pregnancy) is possible only if the potential benefit to the mother outweighs the possible risk to the fetus.

If it is necessary to use the drug during lactation, breastfeeding should be suspended.

The drug should be used with extreme caution in elderly and debilitated patients, because Such patients are more likely to experience side effects (dizziness, drowsiness).

Suprastin should be prescribed with caution simultaneously with sedatives, tranquilizers, analgesics, MAO inhibitors, tricyclic antidepressants, atropine and/or sympatholytics.

During treatment, the consumption of alcoholic beverages should be avoided. Alcohol is harmful when taken simultaneously with any medications.

Each tablet contains 116 mg of lactose monohydrate. This amount may cause undesirable reactions in patients with lactase deficiency or the rare metabolic disorders galactosemia or glucose/galactose malabsorption syndrome.

Impact on the ability to drive vehicles and operate machinery

During the initial, individually determined period of use of Suprastin, driving vehicles and engaging in other potentially hazardous activities that require rapid psychomotor reactions are not allowed. In the process of further treatment, the degree of restrictions is determined depending on the individual tolerability of the drug.

With simultaneous use, Suprastin enhances the effects of sedatives, tranquilizers, analgesics, MAO inhibitors, tricyclic antidepressants, atropine, sympatholytics and ethanol.

When used simultaneously with ototoxic drugs, Suprastin may mask early signs of ototoxicity.

Analogues of the drug Suprastin

Structural analogues of the active substance:

  • Chloropyramine;
  • Chloropyramine-Ferein;
  • Chloropyramine hydrochloride.

Source: http://instrukciya-otzyvy.ru/36-suprastin-po-primeneniyu-analogi-tabletki-ukoly-krapivnica-zud-allergicheskie-zabolevaniya.html

Suprastin's analogs

The drug is very popular in our country, and there are reasons for this - it has a good effect, time-tested and at the same time quite safe (prescribed even to small children). Is there a worthy replacement for it?

The main active ingredient of Suprastin is chloropyramine.

If you need an injection solution, it can often be found in pharmacies under the brand name “Chloropyramine”, at a price lower than the “original”.

Chloropyramine tablets from other manufacturers are sold, although not often. At the time of writing, only 25% of pharmacies had such a product in their assortment. And their cost is approximately two times lower than Suprastin. There are no more complete analogues.

Remember that low price does not mean good quality. Large manufacturers, as a rule, care about their reputation and produce guaranteed quality products, albeit at a higher price.

There are a large number of tablets with a similar effect - antihistamines, here is a list with approximate prices*:

Tablets may differ in contraindications and side effects. Please read the instructions before choosing a replacement!

* - average price among several sellers at the time of monitoring, is not a public offer.

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The drug "Suprastin": analogues. What to choose?

Many people suffer from allergies. Some suffer all year round, while others experience only temporary discomfort when they approach a source that causes unpleasant reactions in them. There are several drugs that can relieve allergic reactions and make life easier. One of them is the drug “Suprastin”. Its analogues are the drugs “Tavegil”, “Fenistil” and others. So, which is better to choose?

Different generations

There are several generations of anti-allergy drugs that differ significantly from each other. The first generation includes potent drugs, which do not act for long and have a severe effect on the body. This is the most popular remedy - “Suprastin”. Its analogues from the same series are the drugs “Tavegil” and “Diphenhydramine”. The second generation includes slower-acting agents. Some medications have side effects. The most popular product from this line was the drug “Fenistil”. The third generation is a little weaker, but these are the easiest and safest drugs in the entire series of anti-allergy drugs. This, in particular, is the drug Zyrtec, which helps in the earliest phase of an allergic reaction.

The drug "Suprastin"

One of the most popular and effective remedies with an antihistamine effect. Helps with swelling and itching, most often used in hospitals when emergency medical assistance is needed. It stops the release of serotonin and histamine, has a calming, almost hypnotic effect, and is a good antispasmodic. The medicine is produced in Hungary and is available in the form of tablets and ampoules. The drug "Suprastin" (its analogues have the same properties) begins to act on average half an hour after entering the body and works for about six hours. True, after seven days, addiction to the drug occurs. This remedy is prescribed for urticaria, hay fever, anaphylactic shock, in the treatment of bronchial asthma, allergic rhinitis and conjunctivitis, eczema, dermatitis and neurodermatitis, for allergies to food, medications and insect bites. It is also used in combination with other medications during the treatment of flu and colds.

Side effects and contraindications

The drug is not indicated for asthma attacks, exacerbation of ulcers, urinary retention, glaucoma, and also together with MAO inhibitors, during pregnancy and lactation. It should not be given to children under one month old and people intolerant to this medicine. Side effects include severe drowsiness, weakness, vomiting, dizziness, dry mouth, and blood pressure problems. Very carefully, the drug "Suprastin" (including its analogues) is given to elderly patients, people with heart, liver, prostate diseases, and those who drive a car or operate any machinery. Under no circumstances should this medicine be mixed with alcoholic beverages.

Means "Tavegil"

When figuring out which is better, Suprastin or Tavegil, you need to consider the following: these are drugs of the same series and of the same generation, and are similar in many ways. The latter is available in tablets and also has a powerful antihistamine and antipruritic effect. It reduces the permeability of capillaries and blood vessels, severe swelling, tumors, and calms (but does not put you to sleep like the drug "Suprastin"). Valid for up to twelve hours. You can drink it for twenty days without fear of addiction. Prescribed for urticaria, fever, dermatoses, eczema, allergies to bites and medications.

Contraindications and special points

The drug "Tavegil" is produced in Italy. It is contraindicated if you are sensitive to it, during pregnancy, lactation, or with lung diseases. It should not be given to children under six years of age. Use with caution for people with diseases of the stomach, bladder, prostate gland, heart and blood vessels, with increased intraocular pressure. In addition, Tavegil causes severe fatigue, weakness, lethargy, drowsiness, dizziness, tremors, problems with coordination of movements, vomiting, constipation, difficulty urinating, blood pressure, and rash. The drug "Tavegil" is much more toxic and heavier than the drug "Suprastin". It has a strong negative effect on kidneys and liver function.

The drug "Fenistil"

This medicine is available in the form of capsules, drops and gel. It is very effective in preventing the development of allergies, reduces swelling that has already formed, and relieves itching. The action occurs within half an hour after taking it for twelve hours, but the gel is felt within a couple of minutes. The drug "Fenistil" is prescribed for urticaria, edema, fever, rhinitis, itchy skin, measles, smallpox and rubella, insect bites, dermatoses, burns, for prevention. When choosing what to buy, the medicine "Fenistil" or "Suprastin", you must first consult a doctor. These are drugs of varying strength and have different indications. When taken, Fenistil may cause mild drowsiness, headaches, nausea, dizziness, rash, spasms, swelling, and breathing problems.

Source: http://www.syl.ru/article/144598/mod_preparat-suprastin-analogi-chto-vyibrat

Suprastin and its analogues: can and should it be replaced?

Every year the number of people susceptible to allergies is growing. The need for special antihistamines is increasing. One of the most famous and widespread antiallergic drugs is Suprastin. Its high efficiency and fairly low price ensure high demand. Most people prefer it as a time-tested drug. But are there other more modern analogues of Suprastin? What can replace this remedy?

Replacing Suprastin: why and why?

Suprastin is a first generation antihistamine produced in Hungary. The main active ingredient is chloropyramine.

Indications for use are various forms of allergies: urticaria, itching, seasonal rhinitis, conjunctivitis, dermatitis, eczema, Quincke's edema, food allergy or allergy from insect bites. In addition to its main use, it is often used for general relief of the patient’s condition.

The sedative property of Suprastin is its main disadvantage - it actively affects the central nervous system and can cause side effects such as drowsiness, dizziness, and general fatigue. Thus, driving a car or active work is sometimes simply impossible. Unpleasant side reactions make you want to learn more about Suprastin and its analogues.

So, what can replace Suprastin? The main analogs of Suprastin come in tablets, but some of them are also available in the form of syrup and special solutions. Below is a list of possible remedies.

Diazolin

Diazolin is a cheap and popular analogue of Suprastin, which has an antiallergic effect and reduces swelling of the mucous membranes. It does not have a strong hypnotic effect, penetrating into the central nervous system only slightly. It has mild anesthetic properties. Used for the combined treatment of bronchial asthma. Unlike its predecessor, it does not help in the treatment of viral diseases. It is not a direct analogue of Suprastin and contains a different active ingredient.

Main active ingredient: mebhydrolin.

Indications for use:

  • may lead to disturbances in the functioning of the gastrointestinal tract;
  • from the central nervous system may cause: dizziness, decreased reaction speed, drowsiness or hyperactivity;
  • Often the use is accompanied by dry mouth.

Contraindicated for children under 3 years of age, people with diseases of the gastrointestinal tract, and women during pregnancy and lactation.

The price of the drug varies from 55–80 rubles.

Chloropyramine

Chloropyramine is an inexpensive drug that blocks histamine receptors. It has sedative properties and a mild antispasmodic effect. The effect occurs after 1–2 hours, the duration of the effect is 4–6 hours. In small doses, it can be used in children from 1 month.

Main active substance: chloropyramine.

  • dermatological diseases: eczema, dermatoses, contact dermatitis, itchy skin;
  • allergic reactions: seasonal allergies, hay fever, conjunctivitis, urticaria.

Since chloropyramine is a direct analogue of Suprastin, it has the same side effects:

  • drowsiness;
  • dizziness;
  • dry mouth;
  • tachycardia;
  • difficulty urinating.

Release form: tablets and solution for injection.

Subrestin

Subrestin is a sedative antihistamine. It has antiallergic, antiemetic and antispasmodic effects. Approved for use in children, in small dosages starting from 1 month.

Main active ingredient: chloropyramine.

Side effects and contraindications are the same as for Suprastin.

Approximate price: 115 rub.

Tavegil

Tavegil is an antiallergic drug, a modern competitor to Suprastin. Fights allergies without causing a calming effect. Reduces swelling, itching and has anesthetic properties. Can be prescribed to children from 6 years of age.

The main active substance of Tavegil: clemastine.

Indications for use:

  • skin diseases: eczema, dermatosis, contact dermatitis;
  • reactions to insect bites and medications;
  • hay fever;
  • anaphylactic shock;
  • allergic swelling;
  • serum sickness;
  • prevention of allergic diseases.
  • dry mouth;
  • nausea, dizziness, headache;
  • hearing and visual impairment;
  • breathing problems;
  • difficulty urinating;
  • cardiopalmus.

Tablets and injections are available commercially. The cost of the drug depends on the packaging, for 10 tablets the approximate price is.

Loratadine

Loratadine belongs to the second generation of antihistamines. It has a rapid and prolonged effect, with no sedative effect. It has virtually no effect on the central nervous system. Adverse reactions are rare: dry mouth or vomiting. Can be used by children from 2 years of age. Do not use during pregnancy or breastfeeding, with caution in case of liver failure.

Main active ingredient: loratadine.

Indications for use:

  • allergic reactions of various origins;
  • dermatological diseases: skin itching, eczema, dermatoses.

With enormous potential, this drug is cheaper than many other drugs: from 35–50 rubles.

Tsetrin

Cetrin is a second generation antihistamine. Reduces the severity of allergic reactions and has an anti-inflammatory effect. It does not affect the functioning of the central nervous system, but its effectiveness is lower than that of Suprastin. Cetrin is prescribed by a doctor as a prophylactic for the treatment of allergies. It can prevent the risk of developing allergic reactions. Suitable for children over 6 years old. Available in syrup and tablets.

Active ingredient: cetirizine.

Main indications for use:

  • seasonal and year-round rhinitis;
  • swelling;
  • hives;
  • skin allergic diseases.

The cost of packing tablets is 10 pcs. — 155–165 rub. syrup price.

The number of available products with a similar spectrum of action is quite large. A cheap or expensive analogue of Suprastin may have the same side effects, while obviously differing in price. Expensive drugs are not necessarily always good. And direct cheap analogues contain the same main component as Suprastin, so you shouldn’t be afraid of them. You need to choose, taking into account specific individual needs, body characteristics and doctor’s recommendations.

Source: http://medanalogi.com/s/suprastin.html

Suprastin - instructions, cheap analogues, which is better, comparison of effectiveness

Suprastin is a drug well known to people suffering from allergies. This medicine is constantly found in home medicine cabinets for allergy sufferers. The main advantages of the drug are low cost and good therapeutic effect. But in pharmacies you can also find analogues of Suprastin. Analogs are cheap. But how much more effective are they than the original?

Chemical composition and dosage forms

Suprastin is a drug that has an antiallergic effect. It belongs to the histamine H1 receptor blockers. The active ingredient is chloropyramine hydrochloride. The medicine is sold in tablet form, as well as in the form of a solution for injections.

The tablets are sealed in blisters of 10 pieces; the package contains two blisters.

Ampoules are sealed in blisters of 5 and 10 pieces. One tablet contains 25 mg of the active substance, 1 ml of solution for intramuscular and intravenous administration contains 20 mg of chloropyramine hydrochloride.

Instructions for use of Suprastin

Indications for use

Suprastin is prescribed for the following diseases and conditions of the body:

  • Allergic rhinitis;
  • Food and drug allergies;
  • Consequences of insect attacks;
  • Conjunctivitis;
  • Eczema;
  • Rashes of various origins;
  • Hives;
  • Allergic dermatosis;
  • Angioedema.

Contraindications for use

You should not use the drug in the following cases:

  • During pregnancy, while breastfeeding;
  • With a lack of lactase in the body, non-acceptance of lactose;
  • In the acute phase of bronchial asthma;
  • In case of intolerance to the components of the drug.

Dosage of the drug in tablet form

Children from three to fourteen years old are usually prescribed 25 mg of the active substance per day, that is, one tablet. Doctors allow children from the age of six to take one and a half tablets. It is advisable to divide the daily dose into two parts, that is, the child should take half a tablet twice a day.

Adults are prescribed 100 mg of medication per day. The daily dose is divided into three doses.

Dosage of the drug in solution form

Intramuscular and intravenous administration of the solution is carried out in the following doses:

  • Infants from one month to one year - 0.25 ml;
  • Children from one to six years old – 0.5 ml;
  • Children from six to fourteen years old – 1 ml;
  • Adults – 2 ml.

Overdose and side effects

It is forbidden to exceed the dose of the medicine recommended in the instructions. The optimal dose is 2 mg per kilogram of human weight. The duration of the therapeutic course is determined only by the doctor. The most commonly observed side effects are:

  • Migraine;
  • Drowsiness;
  • Urge to vomit;
  • Decreased blood pressure;
  • Arrhythmia;
  • Decreased leukocytes in the blood;
  • Tremor, convulsions;
  • Stomach ache;
  • Impaired urination;
  • Glaucoma;
  • Distortion of visual perception;
  • Photodermatitis.

If at least one of the above symptoms appears, you should stop taking the medicine and consult a doctor. In case of severe side effects, the doctor prescribes absorbent medications and gastric lavage to the patient.

Cost of the drug

Suprastin is inexpensive. A package containing 20 tablets costs an average of 130 rubles. A blister with 5 ampoules will cost the buyer approximately 150 rubles.

What are the analogues of suprastin?

Suprastin is a cheap medicine, but many allergy sufferers want to find anti-allergy medicines even cheaper. But the price of therapy is not the only reason for searching for analogues.

  1. Many patients are not satisfied with the chemical composition and side effects of the drug. The big disadvantage of Suprastin is its soporific effect on the body.
  2. The medication reduces the tone of the central nervous system, causing migraines, drowsiness, lethargy, and dizziness. With such side effects, it is impossible to engage in intellectual work, and driving a car is dangerous.

Diazolin or Suprastin – what to choose?

Diazolin is an inexpensive and high-quality analogue of Suprastin. This antiallergic medicine, which reduces swelling of the mucous membranes, has virtually no effect on the nervous system, and therefore does not have a soporific effect. May have a slight anesthetic effect. The drug is sold in the form of tablets and dragees. The active ingredient is mebhydrolin.

Diazolin is used to treat the following diseases:

The drug is often used in the complex therapy of bronchial asthma. When using the medication, the following side effects are observed:

  • Disturbances in the functioning of the digestive tract;
  • Dizziness;
  • Drowsiness or, conversely, agitation;
  • Slowing down reactions to external stimuli;
  • Feeling of dryness in the mouth.

Loratadine or Suprastin – which is better to buy?

Loratadine is a second-generation antihistamine, faster-acting and more effective than Suprastin. It has a weak effect on the nervous system and does not have a soporific effect. The medicine is sold in the form of tablets for oral administration, effervescent tablets, and sweet syrup. The active ingredient is loratadine.

The medication is used to treat the following diseases:

Side effects in rare cases include vomiting and dry mouth. Loratadine is allowed to be taken by children over two years of age. Pregnant women and breastfeeding mothers should not use the drug.

Cetrin or Suprastin - which is cheaper and more effective?

Cetrin is a second generation antihistamine. It significantly weakens the course of the allergic reaction and has an anti-inflammatory effect. Cetrin, unlike Suprastin, does not inhibit the functioning of the nervous system at all. The drug is sold in the form of drops, tablets and sweet syrup. The active substance is cetirizine.

Medicines are prescribed to treat the following diseases:

Tavegil or Suprastin - which is better to buy?

Tavegil is a worthy analogue of Suprastin, a highly effective antiallergic drug. It quickly extinguishes the allergic reaction, relieves swelling, reduces itching, has an anesthetic effect, but does not have a soporific effect. The medicine is sold in tablet form, as well as in the form of a solution for intravenous and intramuscular injections. The active substance is clemastine.

Tavegil is used to treat the following pathologies:

  • Hay fever;
  • Eczema;
  • Dermatosis;
  • Allergies of any origin;
  • Edema;
  • Anaphylactic shock;
  • Consequences of insect attacks.

The drug can be taken by children from the age of six. When treated with Tavegil, the following side effects may occur:

  • Dry mouth;
  • Migraine, dizziness;
  • Nausea;
  • Difficulty breathing;
  • Problems urinating;
  • Tachycardia;
  • Hearing impairment, distortion of visual perception.

A package with ten tablets costs 135–155 rubles, with twenty tablets – 175–200 rubles. Five ampoules will cost the buyer 200–220 rubles.

Suprastin or Zyrtec – what to buy?

Zyrtec is an antiallergic drug that does not produce a soporific effect if the dosage specified in the instructions is followed. The medication is sold in tablet and drop form. The active ingredient is cetirizine dihydrochloride.

The following diseases are treated with the drug:

  • Allergic rhinitis;
  • Conjunctivitis;
  • Hives;
  • Angioedema;
  • Hay fever;
  • Dermatosis.

Pregnant women, breastfeeding mothers, and children under six years of age are not allowed to take the medicine. Also, the medication should not be used by people who have lactose intolerance, glucose-galactose malabsorption syndrome, lactase deficiency in the body, or those suffering from kidney diseases.

Zodak or Suprastin – what to choose?

Zirtek and Zodak are analogues in composition. The active component of these drugs is cetirizine dihydrochloride. Therefore, the effects of the medications are the same. Zyrtec is a Swiss drug, and Zodac is a Czech drug. Zodak is sold in tablet and drop forms. Tablets can be used by children from the age of six, drops - from the age of one. Zodak has a depressing effect on the nervous system, negatively affecting concentration and clarity of consciousness.

Unfortunately, the drug, unlike Suprastin, is not produced in the form of an injection solution, so it cannot be used in severe cases of allergies. Ten tablets cost 120–150 rubles, drops cost 200 rubles.

Fenistil or Suprastin?

Fenistil is a drug often used in pediatrics. The medicine is sold in the form of capsules, gel, drops. The drop form of the medication can be used to treat infants from one month of age. Suprastin is not produced in the form of drops, and this is its disadvantage. The active substance is dimentidene maleate. Fenistil helps cure the following diseases:

  • Hay fever;
  • Allergic rhinitis;
  • Urticaria;
  • Food and drug allergies;
  • Angioedema;
  • Eczema;
  • Consequences of insect attacks;
  • Dermatitis.

Suprastin. They have a quick healing effect, eliminate the rash well, and relieve the burning sensation. . Cheap analogues of Advantan.

Suprastin is also often prescribed for a number of diseases, which includes serum sickness, eczema, atopic dermatitis and rhinitis.

According to statistics from the World Health Organization, 85% of the world's population suffers from allergic reactions of various origins.

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Suprastin. They have a quick healing effect, eliminate the rash well, and relieve the burning sensation. . Cheap analogues of Advantan.

Suprastin is also often prescribed for a number of diseases, which includes serum sickness, eczema, atopic dermatitis and rhinitis.

Source: http://ozude.ru/preparaty/suprastin-analogi-deshevle/

Suprastin: instructions for use

Suprastin tablets represent a clinical and pharmacological group of drugs - H-histamine receptor blockers. They have an antiallergic therapeutic effect and are used to reduce the severity of allergic reactions.

Dosage form, composition

Suprastin tablets are white, round in shape and have a flat-cylindrical surface. The main active ingredient of the drug is chloropyramine, its content in one tablet is 25 mg. It also contains excipients, which include:

  • Potato starch.
  • Stearic acid.
  • Lactose monohydrate.
  • Sodium carboxymethyl starch.
  • Gelatin.
  • Talc.

Suprastin tablets are packaged in blister packs of 10 pieces. The cardboard pack contains 2 blisters with tablets, as well as instructions for use of the medicine.

Therapeutic effects, pharmacokinetics

The main active component of Suprastin tablets, chloropyramine, is a chemically modified derivative of the classic antiallergic compound pyribenzamine due to the addition of chlorine atoms. It blocks H-histamine receptors, due to which they become insensitive to the main mediator of a specific allergic reaction, histamine, produced by some cells in response to the entry of an allergen into the human body, subject to the presence of sensitization (hypersensitivity). This compound also partially blocks M-cholinergic receptors. Due to such physiological effects, several therapeutic actions are realized, namely antiallergic, antiemetic and moderate antispasmodic effects.

After taking the Suprastin tablet orally, the active ingredient is quickly and almost completely absorbed into the blood from the intestinal lumen. It is evenly distributed in tissues and penetrates the structures of the central nervous system through the blood-brain barrier. Chloropyramine is metabolized in the liver to form inactive breakdown products, which are excreted from the body in the urine by the kidneys. The drug is eliminated more quickly in children.

Indications for use

Medical indications for the use of Suprastin tablets are various manifestations of allergies in humans, which include:

  • Skin rash, itching.
  • Urticaria, reminiscent of a nettle burn on the skin.
  • Angioedema of Quincke with a pronounced increase in soft tissue volume and predominant localization in the face and external genitalia.
  • Serum sickness with fever developing after administration of immunobiological drugs.
  • Allergic rhinitis (specific inflammation of the nasal mucosa), which has a year-round or seasonal course.
  • A food or drug allergic reaction of varying severity and localization in the body.
  • Skin itching of various origins.
  • Allergic conjunctivitis is a specific inflammation of the conjunctiva of the eye.
  • Acute or chronic course of eczema with characteristic skin manifestations.
  • Contact dermatitis, the development of which is caused by local contact of the skin with various types of allergens.

The drug is also used to reduce the severity of a specific allergic reaction caused by the ingestion of foreign proteins during bites of various insects.

Contraindications for use

There are several pathological and physiological conditions of the patient’s body that are contraindications for the use of Suprastin tablets, these include:

  • Newborn period of the child (contraindication applies to premature and full-term children).
  • Pregnancy and lactation (breastfeeding) in women.
  • An acute attack of bronchial asthma with the development of paroxysmal cough and shortness of breath.

The drug is used with caution in cases of increased intraocular pressure due to angle-closure glaucoma, deterioration of the functional state of the liver or kidneys, cardiovascular pathology, hyperplasia (increase in volume) of the prostate gland in men, as well as disturbances in the process of urine excretion. The elderly age of the patient requires careful use of this medication. Before starting to use Suprastin tablets, you must ensure that there are no contraindications.

Method of use, dosage

Suprastin tablets are intended for oral (inside) use. They are taken with meals, not chewed and washed down with plenty of water. The average therapeutic dosage for adults is 1 tablet 3-4 times a day, for children aged 6 to 14 years, ½ tablet 3 times a day, for children aged 1 to 6 years, ½ tablet 2 times a day, aged from 1 month to 1 year, ¼ tablet 2-3 times a day (the drug is pre-dissolved in baby formula). The duration of the course of therapy is determined by the disappearance of the manifestations of the allergic reaction. Typically it lasts up to 5 days.

Side effects

While taking Suprastin tablets, it is possible to develop negative pathological reactions provoked by the action of the main active component of the drug on the part of various organs and systems:

  • Digestive system - pain in the abdomen, mainly in its upper parts, nausea accompanied by periodic vomiting, increased or decreased appetite up to its complete loss, diarrhea or constipation, dry mouth.
  • Nervous system – increased fatigue, periodic dizziness, trembling (tremor) of the hands, drowsiness, nervous agitation.
  • Cardiovascular system - decreased blood pressure, irregular heartbeat (arrhythmia), increased heart rate (tachycardia).
  • Urinary system – difficulty urinating.
  • Blood and red bone marrow – decrease in the number of leukocytes (leukopenia), granulocytes (agranulocytosis) in the blood.
  • Musculoskeletal system – muscle weakness (myasthenia gravis).
  • Sense organs – increased intraocular pressure.
  • Skin and its appendages – increased sensitivity to light (photosensitivity).

The appearance of signs of negative side reactions is a reason to stop taking Suprastin tablets and consult a doctor, who will determine the possibility of further use of the drug.

Special Recommendations

Before starting to take Suprastin tablets, it is important to carefully read the instructions for the drug. There are several special recommendations regarding the use of the drug that are worth paying attention to, these include:

  • Pathological processes localized in the liver or kidneys and accompanied by a decrease in the functional activity of organs require a reduction in the dosage of the drug.
  • With concomitant reflux esophagitis in a patient, taking Suprastin tablets at night can provoke an increase in the manifestations of this pathological process in the form of heartburn.
  • During the course of treatment with this drug, you should avoid drinking alcohol, as it may increase its inhibitory effect on the functional activity of the nervous system.
  • In patients with impaired digestion and absorption of certain carbohydrates in the intestine, dyspepsia may develop, which is provoked by lactose, which is part of the tablets.
  • The combined use of this drug with ototoxic drugs may mask the manifestations of their ototoxicity.
  • The drug can enhance the inhibitory effect on the structures of the nervous system of antidepressants, tranquilizers, M-anticholinergics, analgesics, and monoamine oxidase (MAO) enzyme inhibitors.
  • The active component of this drug can cause drowsiness and depression of the functional activity of the nervous system, therefore it is not recommended to perform potentially dangerous types of work while taking it, especially in the first days of the course of therapy.

In the pharmacy chain, Suprastin tablets are available without a prescription. If you have doubts about their use, this is grounds for contacting a medical specialist.

Exceeding the dosage

Significantly exceeding the recommended therapeutic dose of Suprastin tablets causes the development of hallucinations, severe anxiety, impaired coordination of movements, anxiety, dry mouth, dilated pupils, increased heart rate, redness of the facial skin, convulsions, disturbances of consciousness up to coma. In this case, gastric and intestinal lavage is carried out, intestinal sorbents (activated carbon) are taken, as well as symptomatic therapy in a medical hospital under the control of indicators of the functional activity of vital organs and systems.

Analogs of Suprastin tablets

A drug similar in structure and therapeutic effect to Suprastin tablets is Chloropyramine.

Storage rules

The shelf life of Suprastin tablets is 5 years. They must be stored in their entire packaging, in a dark, dry place, out of reach of children, at an air temperature no higher than +25° C.

Suprastin tablets price

The average cost of Suprastin tablets in Moscow pharmacies varies within rubles.

Source: http://bezboleznej.ru/suprastin

"Suprastin": instructions for use, price, analogues

Despite the development of second-generation antiallergic drugs, previous drugs will remain widely used in clinical allergology. The classic representative of the first generation antihistamines is Suprastin.

Description of the drug

The drug can be presented in the following form:

  • The tablets are disc-shaped, grayish-white or pure white. Sometimes there is a slight specific aroma. Each pill is marked “suprastin” and has a chamfer.
  • A solution synthesized for intramuscular or intravenous administration. Aqueous, colorless, transparent liquid. A faint specific aroma is observed. The ampoules are marked with a red code ring, the break point.

Pharmacokinetics and pharmacodynamics:

  • The dynamic and kinetic characteristics of the drug suggest complete absorption of the active substance from the digestive tract.
  • “Suprastin” spreads well throughout the body, penetrating the central nervous system.
  • Active metabolites are formed in the liver.
  • Excretion is carried out by the kidneys.
  • In childhood, the elimination of the drug occurs more intensely.
  • The primary therapeutic effect appears after 15 minutes. after internal reception.
  • The therapeutic effect lasts more than three hours.

If you are one of those people who try to be treated with folk remedies, then this article will be interesting to you.

The medicinal effect of the drug can be described as follows:

  • First generation antiallergic drug, histamine receptor blocker.
  • The medication has anticholinergic and antihistamine effects against the background of moderate antispasmodic and peripheral activity.

The chemical composition of the drug is indicated in the tabular data.

  • “Suprastin”, tablet form, cardboard packs with instructions included, foil blisters/polymer jars. The cost of package No. 20 is 110 rubles.
  • “Suprastin”, ampoule form, cardboard packs with instructions included, foil blisters. The cost of packaging product No. 5 is 153 rubles.

Pharmacy conditions, storage rules, expiration date:

  • Available over-the-counter from pharmacy chains for tablet form. Suprastin ampoule is available by prescription.
  • Storage must be provided under special conditions: a place with moderate humidity, isolated from sunlight and access to children. The temperature norm is no higher than 25 degrees.
  • The drug maintains stable pharmacological characteristics for 5 years.

Interaction with other drugs

When using the drug, you must familiarize yourself with the pharmacological compatibility standards:

  • The medication greatly enhances the effect of drugs intended for anesthesia and sedative drugs.
  • "Suprastin" is not recommended to be taken together with tranquilizers, MAO inhibitors, and analgesics.
  • When taken simultaneously with sympatholytics, Atropine, and tricyclic antidepressants, the pharmacological action of the latter is accelerated.

Indications. Contraindications. Overdose

The drug is taken strictly according to indications:

  • Urticaria is a disease affecting the skin, primarily caused by allergies (allergies).
  • Quincke's edema (angioneurotic).
  • Rhinitis of allergic origin, occurring in a chronic or seasonal form (Allergic rhinitis and otitis media).
  • Contact, atopic dermatitis and photodermatosis are a type of allergy that occurs with significant skin lesions.
  • Conjunctivitis (inflammation of the mucous membrane of the eyes).
  • Itching covering the skin.
  • Allergy to medications – caused by taking medications.
  • Food allergy is the body's reaction to a food irritant.
  • Negative reaction to insect bites.

The drug should not be used if the following conditions are detected:

  • Increased sensitization to the components of Suprastin.
  • Bronchial asthma, during acute attacks.
  • Cautious use - in case of detection of prostate hyperplasia, glaucoma (in closed-angle form), diseases of the heart, blood vessels, liver, kidneys.

The intake and dosage of the medication must comply with the following principles:

  • The tableted drug is intended for oral administration.
  • It is recommended to take the product with food, accompanied by a moderate amount of liquid, preferably water.
  • Adult patients are prescribed 25 mg, which corresponds to one pill 3-4 times a day. The daily value is 75.0-100.0 mg.
  • The ampoule form is used in acute cases under professional medical supervision.
  • In adults, 1-2 ml of the drug is prescribed intramuscularly, which corresponds to 1-2 ampoules.

Use of the drug in special groups of patients

  • Persons suffering from exhaustion, elderly patients. The medication is prescribed with caution, with the correct dose calculation, since Suprastin may lead to the development of unwanted side effects.
  • Persons with acute liver failure - it is possible to adjust the dose downwards, which is due to a reduction in metabolism.
  • Persons with acute liver failure. Active metabolites are excreted by the kidneys, so a downward dose adjustment is required.
Taking the medication may cause a response from the body:
  • Hallucinations.
  • Anxiety.
  • Ataxia is poor coordination of movements.
  • Insufficient coordination of movements.
  • Atheosis – slow, tonic spasms of the limbs.
  • Convulsive states.
  • Redness of the face, fever.
  • Excitement leading to depression and coma.
  • In childhood, fixation of dilated pupils, dry mouth, anxiety, agitation, fever, coma, tachycardia, and reddening of the cheeks are observed.

Side effects and special instructions

Signs that determine side effects last a short period and are quickly minimized when the drug is discontinued:

  • Drowsiness, excessive fatigue, tremors, overexcitation, euphoria, headaches.
  • Discomfort in the abdominal area, vomiting and nausea, stool instability, diarrhea, changes in appetite.
  • Tachycardia, arrhythmia, low blood pressure.
  • Leukopenia is a decrease in the number of leukocytes in the blood.
  • Agranulocytosis is a pathological condition accompanied by a decrease in the level of leukocytes, including due to granulocytes.
  • Difficulty urinating.
  • Weakness spreading through the muscles.
  • Sensitivity to light.
  • The occurrence of high intraocular pressure.

The use of the medication should be accompanied by the study of additional instructions:

  • Primary signs of ototoxicity can be masked by taking Suprastin (together with ototoxic drugs).
  • Dose adjustment is mandatory if the patient suffers from liver and kidney diseases.
  • Symptoms of reflux esophagitis syndrome may increase if Suprastin is taken at night.
  • The drug cannot be combined with alcohol or ethanol.
  • The medication contains lactose, which is important to consider when treating patients with lactase deficiency.
  • At the early stage of therapy, you should refrain from driving vehicles and potentially dangerous types of work. The restriction can be lifted by the attending physician, taking into account the patient’s condition.
  • For women who are breastfeeding, taking the drug forces them to stop lactation.
  • During pregnancy, the medication is prescribed only if the expected benefit outweighs the expected risk to the fetus.

Use of the drug in childhood

  • The dosage can be gradually increased if the drug is well tolerated.
  • The daily rate should not exceed 2.0 mg/kg.
  • The tablet is crushed into powder and presented to the child along with baby food.
  • The drug is not prescribed to newborn children.

Suprastin analogues in tablets

Drugs with a similar spectrum of action are listed below.

The drug blocks the development of allergic reactions and facilitates their course. The dosage is calculated individually.

  • The drug is used in the treatment of serum sickness.
  • The medication is a derivative of ethylenediamine.

The cost of the product is 126 rubles.

The medication has an antipruritic effect and relieves inflammatory reactions. The dosage is calculated individually.

  • The drug is available in the form of powdered substances.

The cost of the product is 87 rubles.

Reviews

I always drink Suprastin for any manifestations of food allergies. This great remedy always comes to the rescue when you eat something wrong.

I take the drug for preventive purposes, as I suffer from year-round allergies. The drug is well tolerated and is highly effective even during long-term therapy.

After I found out why Suprastin also helps, I started taking it for prevention.

"Suprastin" is an effective first-generation antihistamine that allows you to successfully stop any manifestations of allergies.

Source: http://provitaminki.com/zdorovie/allergiya/suprastin.html