Suprastin what is it for?

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What does Suprastin help with?

Suprastin is one of the most effective antihistamines, which helps to quickly relieve any allergic reaction.

The main active ingredient of Suprastin is chloropyramine, which has pronounced antiallergic properties.

Table of contents:

Also, this drug exhibits minor antiemetic and antispasmodic effects.

Suprastin also helps well with various allergic reactions in children (urticaria, allergic rhinitis, itchy skin, conjunctivitis, etc.), and it can be taken from almost 1 month of life.

The medicinal (therapeutic) effect after internal administration of Suprastin develops within a minute, and its maximum effect begins approximately after a minute.

Main indications for use of Suprastin:

  • severe or moderate skin itching;
  • food or drug allergies;
  • contact dermatitis;
  • hives;
  • serum sickness;
  • allergic rash;
  • seasonal rhinitis;
  • swelling;
  • acute or chronic form of eczema;
  • allergic manifestations to insect bites;
  • Quincke's edema;
  • anaphylactic shock.

Attention: before long-term use of Suprastin, it is recommended to consult a doctor!

The drug is available in the form of tablets and solutions for intramuscular administration.

How to take Suprastin?

The daily dose of Suprastin for adults is 1 t. 2-3 r. daily after meals with plenty of water. The minimum interval between doses should be at least 4-5 hours.

For children from 1 to 12 months. the medicinal dose is ¼ t. 2-3 r. in a day. From 1 to 6 years it is recommended to give 1/3 t. 2-3 r. for a day. It is advisable for children from 7 to 15 years old to take ½ t. 2-3 r. per day after meals. In more severe situations, Suprastin is recommended to be administered intramuscularly in a total dose of 1-2 ml. (for adults).

It is strictly not recommended to exceed the required dose of the drug, so as not to provoke a possible overdose, which can mainly be manifested by nausea, dizziness, vomiting, diarrhea, dry mouth, drowsiness and other symptoms.

Contraindications to the use of Suprastin

  • not recommended for use in children under 1 month of age;
  • attack of bronchial asthma;
  • pregnancy;
  • impaired functioning of the kidneys and liver;
  • lactation period (breastfeeding);
  • BPH;
  • glaucoma.

Side effects of Suprastin

As a rule, after taking Suprastin, side effects can extremely rarely occur, the most common of which are:

  • general weakness, lethargy, fatigue;
  • nausea;
  • decreased appetite;
  • diarrhea;
  • dry mouth;
  • dizziness;
  • constipation;
  • heartbeat disturbance (bradycardia or tachycardia);
  • intestinal colic;
  • arterial hypertension (high blood pressure);
  • urinary disturbance.

If any of the above side effects develop, you must completely stop further use of the drug, and also be sure to consult a doctor!

In this article, we looked at what Suprastin helps with, as well as how to take it correctly.

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Remember, self-medication is dangerous to your health! Consult your doctor

Source: http://in4health.ru/ot-chego-pomogaet-suprastin.html

Suprastin - instructions for use: price, analogues and dosage for children, adults and during pregnancy

Suprastin is a prominent representative of the first generation of antihistamines, the mechanism of use of which is aimed at blocking histamine receptors and providing an antispasmodic effect. Numerous studies that have been conducted on chloropyramine have shown that Suprastin is very effective in the treatment of hay fever and other allergic pathologies.

Despite the emergence of the latest generation of drugs with a limited list of side effects, Suprastin is still used when an immediate effect is needed. 15 minutes pass and the first signs of the action of the antiallergic drug are already noticeable. However, do not forget that self-medication can lead to undesirable results. Suprastin can be self-prescribed once before the doctor arrives, only in an emergency. Or if you are sure that the child is really having an allergy attack and has already had such signs before and the drug has already been prescribed.

How does suprastin work?

In the treatment of allergic reactions, drugs that affect histamine metabolism (antihistamines) are used. The action of suprastin in allergies is primarily aimed at suppressing the activity of histamine. Suprastin blocks histamine receptors (H1), thus preventing the appearance of signs and symptoms of allergies. In addition, suprastin has a pronounced antipruritic effect.

After taking Suprastin orally, the drug is quickly and completely absorbed into the blood from the intestines. The maximum concentration of the drug is reached 2 hours after application. As a rule, suprastin distributes well in the human body (penetrates the brain). The drug is excreted through the kidneys (in case of renal failure, the dose of the drug should be reduced).

Pharmacodynamics

Chloropyramine, a chlorinated analogue of tripelenamine (pyribenzamine), is a classic antihistamine that belongs to the group of ethylenediamine antihistamines. A blocker of H1-histamine receptors, has an antihistamine and m-anticholinergic effect, has an antiemetic effect, moderate antispasmodic and peripheral anticholinergic activity.

Pharmacokinetics

When taken orally, it is almost completely absorbed from the gastrointestinal tract (GIT). The therapeutic effect of chloropyramine develops within 15–30 minutes after oral administration, reaches a maximum within the first hour after administration and lasts at least 3–6 hours. Well distributed throughout the body, including the central nervous system (CNS). Intensively metabolized in the liver. It is excreted mainly by the kidneys. In children, drug elimination occurs faster than in adult patients.

Indications for suprastin

  • hives;
  • angioedema (Quincke's edema);
  • serum sickness;
  • seasonal and year-round allergic rhinitis;
  • conjunctivitis;
  • contact dermatitis;
  • skin itching;
  • acute and chronic eczema;
  • atopic dermatitis;
  • food and drug allergies;
  • allergic reactions to insect bites.

Contraindications

  • hypersensitivity to the components of the drug;
  • acute attack of bronchial asthma;
  • newborn babies (full-term and premature);
  • pregnancy;
  • lactation period.
  • angle-closure glaucoma;
  • urinary retention;
  • prostatic hyperplasia;
  • liver and/or kidney dysfunction;
  • cardiovascular diseases;
  • elderly patients.

Method of application and dosage of suprastin

The tablets are taken orally during meals, without chewing and with a sufficient amount of water.

For adults

Prescribe 1 tablet 3-4 times a day (75-100 mg per day).

For children

  • at the age of 1 to 12 months - 1/4 tablet (6.5 mg) 2-3 times a day (ground to powder along with baby food);
  • At the age of 1 to 6 years - 1/4 tablet 3 times a day or 1/2 tablet 2 times a day;
  • At the age of 6 to 14 years - 1/2 tablet (12.5 mg) 2-3 times a day.

The dose can be gradually increased if the patient has no side effects, but the maximum dose should never exceed 2 mg/kg body weight.

Special patient groups

Elderly, debilitated patients: the use of the drug Suprastin requires special caution, because in these patients, antihistamines are more likely to cause side effects (dizziness, drowsiness).

Patients with impaired liver function: a dose reduction may be required due to a decrease in the metabolism of the active component of the drug in liver diseases.

Patients with impaired renal function: a change in the dosage regimen and a dose reduction may be required due to the fact that the active component is mainly excreted through the kidneys.

How long can you take Suprastin

The course of treatment with Suprastin is prescribed by a doctor and is selected individually for each patient depending on the course of the disease and its complexity.

Use of suprastin during pregnancy

There have been no adequate and well-controlled studies of the use of antihistamines during pregnancy. Therefore, the use of the drug in pregnant women (especially in the first trimester and the last month of pregnancy) is possible only if the potential benefit to the mother outweighs the possible risk to the fetus.

If it is necessary to use the drug during lactation, breastfeeding should be suspended.

The use of suprastin in childhood

It can be used according to indications and in doses taking into account the patient’s age. The drug is not prescribed to newborns (including premature infants). The medicine is recommended for children starting from 1 month of life. The course and frequency of use directly depend on the pathological process. In case of mild manifestations of an allergic reaction, the drug can be given to the child no more than 1 time per day. And if the allergy occurs in a complex form, then you can take the drug 3 times a day.

Parents should remember that a child may have a completely atypical reaction to the drug Suprastin in the form of hyperexcitability, anxiety and insomnia. The course of treatment for children with Suprastin cannot last more than 7 days; if during this period of time the signs of allergy have not disappeared, then you need to seek help from a doctor.

Side effects

Side effects, as a rule, occur extremely rarely, are temporary, and disappear after discontinuation of the drug.

  • From the central nervous system: drowsiness, fatigue, dizziness, nervous excitement, tremor, headache, euphoria.
  • From the gastrointestinal tract: abdominal discomfort, dry mouth, nausea, vomiting, diarrhea, constipation, lack or increased appetite, pain in the upper abdomen.
  • From the cardiovascular system: decreased blood pressure, tachycardia, arrhythmia. A direct connection between these side effects and the use of the drug has not always been established.
  • From the hematopoietic system: very rarely: leukopenia, agranulocytosis.

Other: difficulty urinating, muscle weakness, increased intraocular pressure, photosensitivity.

Overdose

Symptoms

  • hallucinations;
  • anxiety;
  • ataxia;
  • impaired coordination of movements;
  • athetosis;
  • convulsions.

In young children, agitation, anxiety, dry mouth, fixed dilated pupils, facial flushing, sinus tachycardia, urinary retention, fever, coma.

In adults, fever and facial redness are observed intermittently, after a period of excitement followed by convulsions and post-convulsant depression, coma.

Treatment

In the period up to 12 hours after taking the drug orally, gastric lavage is necessary (it should be taken into account that gastric emptying is prevented by the anticholinergic effect of the drug). The use of activated carbon is also indicated. Monitoring of blood pressure and breathing parameters is necessary. Symptomatic therapy. Resuscitation measures. A specific antidote is not known.

Interaction with other drugs

The drug should be used with caution with sedatives, tranquilizers, analgesics, MAO inhibitors, tricyclic antidepressants, atropine and/or sympatholytics, since the effects of these drugs may be enhanced when used simultaneously.

Interaction of suprastin with alcohol

Suprastin tends to enhance the effect of ethyl alcohol on the central nervous system. During the course of therapy, you should abstain from any alcohol (including medicinal tinctures).

Special instructions for use

Each tablet contains 116 mg of lactose monohydrate. This amount may cause undesirable reactions in patients with lactose deficiency or rare metabolic disorders - galactosemia or glucose/galactose malabsorption syndrome.

When combined with ototoxic drugs, Suprastin can mask early signs of ototoxicity.

Diseases of the liver and kidneys may require a change (reduction) in the dose of the drug, and therefore the patient should inform the doctor about the presence of

Transport and machinery management

The drug, especially in the initial period of treatment, may cause drowsiness, fatigue and dizziness. Therefore, in the initial period, the duration of which is determined individually, driving vehicles or performing work associated with an increased risk of accidents is prohibited. After this, the degree of restriction on driving vehicles and operating machinery must be determined by the doctor individually for each patient.

Release form

Tablets 25 mg. 20 tablets in brown glass bottles with PE caps. The bottle is packaged in a cardboard box along with instructions for medical use. Or 10 tablets per blister. 2 blisters are packed in a cardboard box along with instructions for medical use.

In addition to the standard pack, in pharmacies there is a variety in the form of ampoules containing 20 mg of chloropyramine hydrochloride. It is sold in packs of 5 ampoules and contains, in addition to the active substance, water for injection.

A solution for intravenous and intramuscular administration is used when there is an urgent need to relieve allergy symptoms - Quincke's edema, suffocation or convulsions. In such cases, the solution is administered intravenously for immediate action. To use at home, you must have skills in intravenous injections for children.

Storage conditions

At a temperature of 15–25 °C, out of the reach of children.

Best before date

5 years. Do not use after the date indicated on the package.

Conditions for dispensing from pharmacies

Price for suprastin

  • tablets 20 pcs. in packaging - from 110 rubles;
  • solution of 10 ampoules per package – from 150 rubles.

Suprastin analogues

Today, there are a large number of antihistamines that help effectively combat the body’s allergic reactions to any of the existing allergens, the most common:

Suprastin or tavegil

What is better to take during allergies - Suprastin or Tavegil? These medications belong to one group of drugs – antihistamines. The main indication for both Suprastin and Tavegil are allergic diseases of various natures.

But what is better – Tavegil or Suprastin? The main difference between these drugs is the manufacturer: Suprastin is a domestic medicine, Tavegil is a foreign one. Unlike Suprastin, Tavegil is prescribed to children over six years of age.

The effectiveness of both drugs is quite high. Both drugs belong to the first generation of antiallergic drugs. The basis of Tavegil is the substance clemastine, and Suprastin is chloropyramine.

Suprastin has a significant side effect: severe drowsiness. Tavegil is devoid of this side effect, which distinguishes it favorably from Suprastin. However, Tavegil has a much wider range of contraindications and side effects.

Suprastin or Cetrin

Cetrin (cetirizine hydrochloride) is a 2nd generation drug that is a highly selective antagonist of H1-type histamine receptors. The drug has 2 release forms - tablets, which are used in patients over 6 years of age, and syrup, which is prescribed from 2 years of age.

Cetirizine hydrochloride is practically not biotransformed in the body; the rate of its elimination is related to the functional state of the kidneys. A special feature of the drug is its ability to penetrate well into the skin, which makes Cetrin especially effective for skin manifestations of allergies.

The drug does not have a proarrhythmic effect, which has been proven in preclinical and clinical studies. This means that the use of Cetrin is much less likely to be accompanied by the development of adverse reactions than the use of 1st generation products. Moreover, the degree of expression of the latter is also less than that of Suprastin.

If we talk about antiallergic activity, then Suprastin is considered a somewhat stronger remedy.

Questions and answers on the topic "Suprastin"

Question: Hello. Today we were given vaccinations (hepatitis B, polio, diphtheria, whooping cough and tetanus), they told us to drink Suprastin 1/4 at home before meals, but they didn’t tell us how many times a day to give or for how long to take it. My son is 4 months old. Do I need to give suprastin and how many times?

Source: http://www.diagnos-online.ru/lekarstvennye-preparaty/suprastin.html

Suprastin: instructions for use

Suprastin tablets represent a clinical and pharmacological group of drugs - H-histamine receptor blockers. They have an antiallergic therapeutic effect and are used to reduce the severity of allergic reactions.

Dosage form, composition

Suprastin tablets are white, round in shape and have a flat-cylindrical surface. The main active ingredient of the drug is chloropyramine, its content in one tablet is 25 mg. It also contains excipients, which include:

  • Potato starch.
  • Stearic acid.
  • Lactose monohydrate.
  • Sodium carboxymethyl starch.
  • Gelatin.
  • Talc.

Suprastin tablets are packaged in blister packs of 10 pieces. The cardboard pack contains 2 blisters with tablets, as well as instructions for use of the medicine.

Therapeutic effects, pharmacokinetics

The main active component of Suprastin tablets, chloropyramine, is a chemically modified derivative of the classic antiallergic compound pyribenzamine due to the addition of chlorine atoms. It blocks H-histamine receptors, due to which they become insensitive to the main mediator of a specific allergic reaction, histamine, produced by some cells in response to the entry of an allergen into the human body, subject to the presence of sensitization (hypersensitivity). This compound also partially blocks M-cholinergic receptors. Due to such physiological effects, several therapeutic actions are realized, namely antiallergic, antiemetic and moderate antispasmodic effects.

After taking the Suprastin tablet orally, the active ingredient is quickly and almost completely absorbed into the blood from the intestinal lumen. It is evenly distributed in tissues and penetrates the structures of the central nervous system through the blood-brain barrier. Chloropyramine is metabolized in the liver to form inactive breakdown products, which are excreted from the body in the urine by the kidneys. The drug is eliminated more quickly in children.

Indications for use

Medical indications for the use of Suprastin tablets are various manifestations of allergies in humans, which include:

  • Skin rash, itching.
  • Urticaria, reminiscent of a nettle burn on the skin.
  • Angioedema of Quincke with a pronounced increase in soft tissue volume and predominant localization in the face and external genitalia.
  • Serum sickness with fever developing after administration of immunobiological drugs.
  • Allergic rhinitis (specific inflammation of the nasal mucosa), which has a year-round or seasonal course.
  • A food or drug allergic reaction of varying severity and localization in the body.
  • Skin itching of various origins.
  • Allergic conjunctivitis is a specific inflammation of the conjunctiva of the eye.
  • Acute or chronic course of eczema with characteristic skin manifestations.
  • Contact dermatitis, the development of which is caused by local contact of the skin with various types of allergens.

The drug is also used to reduce the severity of a specific allergic reaction caused by the ingestion of foreign proteins during bites of various insects.

Contraindications for use

There are several pathological and physiological conditions of the patient’s body that are contraindications for the use of Suprastin tablets, these include:

  • Newborn period of the child (contraindication applies to premature and full-term children).
  • Pregnancy and lactation (breastfeeding) in women.
  • An acute attack of bronchial asthma with the development of paroxysmal cough and shortness of breath.

The drug is used with caution in cases of increased intraocular pressure due to angle-closure glaucoma, deterioration of the functional state of the liver or kidneys, cardiovascular pathology, hyperplasia (increase in volume) of the prostate gland in men, as well as disturbances in the process of urine excretion. The elderly age of the patient requires careful use of this medication. Before starting to use Suprastin tablets, you must ensure that there are no contraindications.

Method of use, dosage

Suprastin tablets are intended for oral (inside) use. They are taken with meals, not chewed and washed down with plenty of water. The average therapeutic dosage for adults is 1 tablet 3-4 times a day, for children aged 6 to 14 years, ½ tablet 3 times a day, for children aged 1 to 6 years, ½ tablet 2 times a day, aged from 1 month to 1 year, ¼ tablet 2-3 times a day (the drug is pre-dissolved in baby formula). The duration of the course of therapy is determined by the disappearance of the manifestations of the allergic reaction. Typically it lasts up to 5 days.

Side effects

While taking Suprastin tablets, it is possible to develop negative pathological reactions provoked by the action of the main active component of the drug on the part of various organs and systems:

  • Digestive system - pain in the abdomen, mainly in its upper parts, nausea accompanied by periodic vomiting, increased or decreased appetite up to its complete loss, diarrhea or constipation, dry mouth.
  • Nervous system – increased fatigue, periodic dizziness, trembling (tremor) of the hands, drowsiness, nervous agitation.
  • Cardiovascular system - decreased blood pressure, irregular heartbeat (arrhythmia), increased heart rate (tachycardia).
  • Urinary system – difficulty urinating.
  • Blood and red bone marrow – decrease in the number of leukocytes (leukopenia), granulocytes (agranulocytosis) in the blood.
  • Musculoskeletal system – muscle weakness (myasthenia gravis).
  • Sense organs – increased intraocular pressure.
  • Skin and its appendages – increased sensitivity to light (photosensitivity).

The appearance of signs of negative side reactions is a reason to stop taking Suprastin tablets and consult a doctor, who will determine the possibility of further use of the drug.

Special Recommendations

Before starting to take Suprastin tablets, it is important to carefully read the instructions for the drug. There are several special recommendations regarding the use of the drug that are worth paying attention to, these include:

  • Pathological processes localized in the liver or kidneys and accompanied by a decrease in the functional activity of organs require a reduction in the dosage of the drug.
  • With concomitant reflux esophagitis in a patient, taking Suprastin tablets at night can provoke an increase in the manifestations of this pathological process in the form of heartburn.
  • During the course of treatment with this drug, you should avoid drinking alcohol, as it may increase its inhibitory effect on the functional activity of the nervous system.
  • In patients with impaired digestion and absorption of certain carbohydrates in the intestine, dyspepsia may develop, which is provoked by lactose, which is part of the tablets.
  • The combined use of this drug with ototoxic drugs may mask the manifestations of their ototoxicity.
  • The drug can enhance the inhibitory effect on the structures of the nervous system of antidepressants, tranquilizers, M-anticholinergics, analgesics, and monoamine oxidase (MAO) enzyme inhibitors.
  • The active component of this drug can cause drowsiness and depression of the functional activity of the nervous system, therefore it is not recommended to perform potentially dangerous types of work while taking it, especially in the first days of the course of therapy.

In the pharmacy chain, Suprastin tablets are available without a prescription. If you have doubts about their use, this is grounds for contacting a medical specialist.

Exceeding the dosage

Significantly exceeding the recommended therapeutic dose of Suprastin tablets causes the development of hallucinations, severe anxiety, impaired coordination of movements, anxiety, dry mouth, dilated pupils, increased heart rate, redness of the facial skin, convulsions, disturbances of consciousness up to coma. In this case, gastric and intestinal lavage is carried out, intestinal sorbents (activated carbon) are taken, as well as symptomatic therapy in a medical hospital under the control of indicators of the functional activity of vital organs and systems.

Analogs of Suprastin tablets

A drug similar in structure and therapeutic effect to Suprastin tablets is Chloropyramine.

Storage rules

The shelf life of Suprastin tablets is 5 years. They must be stored in their entire packaging, in a dark, dry place, out of reach of children, at an air temperature no higher than +25° C.

Suprastin tablets price

The average cost of Suprastin tablets in Moscow pharmacies varies within rubles.

Source: http://bezboleznej.ru/suprastin

What is Suprastin medicine for?

Suprastin tablets are an antihistamine that is used to relieve allergic symptoms. This medicine has a number of contraindications and can cause side effects, so it should be taken only as prescribed by a doctor.

Composition and form

Suprastin can be purchased in pharmacy chains in tablet form and in the form of an aqueous solution intended for intramuscular or intravenous injection. When treating allergic pathologies, specialists most often use tablets of this medication, which have a round shape, white color and are packaged in 10 pieces in special blisters. The active substance in this medication is chloropyramine hydrochloride, the amount of which in one tablet is 25 mg. The drug in the form of a solution is needed for those patients who have an acute form of allergy.

What does Suprastin treat?

The instructions that come with the medicine indicate what Suprastin is used for and what pharmacological effect it has on the body of allergy sufferers. This medication has a pronounced effect:

  • antipruritic;
  • antihistamine;
  • decongestant;
  • anti-inflammatory;
  • antispasmodic.

After taking the medicine, the patient’s body blocks the production of proteins, which begin to form immediately after contact with allergens. The maximum therapeutic effect after taking a Suprastin tablet is achieved after 2 hours, while the therapeutic effect will last for 8 hours.

What should you take Suprastin for?

People should read the instructions carefully to find out what this medication is used for. The manufacturer indicates that the drug will have a therapeutic effect in the presence of the following pathologies:
  1. Hay fever.
  2. Urticaria.
  3. Sinusitis.
  4. Quincke's edema.
  5. Serum pathology.
  6. Rhinitis or conjunctivitis of allergic etiology.
  7. Asthma.
  8. Otitov.
  9. Dermatoses (various types).
  10. Skin rashes.
  11. Eczema.
  12. Fevers.
  13. Animal hair intolerance.
  14. Dermatitis.
  15. Insect bites.

Rules of application

In tablet form, this drug should be used if indicated and after receiving an appropriate prescription from an allergist. If the patient has an acute form of an allergic reaction, then Suprastin should be replaced with a more effective medication. The tablets should be taken after meals. The dosage directly depends on the severity of allergic symptoms, the age category of the patient and the characteristics of his body.

Single dose (maximum dose 100 mg per day)

Teenagers from 14 years old

In acute forms of allergies, adults are administered the drug intramuscularly or intravenously.

Contraindications, side effects

The manufacturer's instructions describe all contraindications to the use of Suprastin. Before starting therapy, patients should study it carefully to prevent the development of adverse reactions.

It is not recommended to take this drug if you have the following pathologies:

  1. Women who are pregnant and during lactation.
  2. In case of individual intolerance to the components of the medication.
  3. During an asthma attack.
  4. With urinary retention.
  5. For acute heart attack and arrhythmia.
  6. In the presence of ulcerative pathology in the gastrointestinal tract.
  7. If you have glaucoma.
  8. When undergoing therapy that involves MAO inhibitors.
  9. In the presence of prostate hyperplasia.

Some patients may develop side effects while taking Suprastin:

  1. Tremors and convulsions appear.
  2. The pressure decreases.
  3. Dizziness begins.
  4. Insomnia appears.
  5. Tachycardia develops.
  6. The mucous membranes in the mouth dry out.
  7. The processes of defecation are disrupted.
  8. Nervous excitability increases.
  9. A skin rash and severe itching appears.

Features of the drug use

When conducting Suprastin therapy, patients should follow the following recommendations:

  1. It is prohibited to drink alcoholic beverages during treatment. This is due to the fact that such a combination will cause a serious blow to the patient’s central nervous system. The patient may lose control of himself and may develop irreversible processes in the liver. Pathological reactions will also occur in the stomach, brain and intestines. When combining alcohol with the drug, the side effects will increase several times.
  2. When undergoing Suprastin therapy, the patient should not drive a vehicle, as the drug causes drowsiness and dulls the reaction. Also during this period you should not perform responsible work that requires high concentration.

Use of Suprastin in the treatment of children

Currently, the manufacturer does not produce a drug intended specifically for children. Despite this, specialists quite successfully use Suprastin in therapy for young allergy sufferers. For such patients, the dosage is determined individually based on the following indicators: age and weight. Suprastin should not be given to newborn babies, as well as infants in the first month of life. In other cases, the following dosages are used:

Children under 1 year

Children from 1 year to 6 years

2-3 times a day

Children under 14 years old

If the baby cannot swallow the tablet, parents should grind it into powder and then dilute it in a tablespoon of water. For infants, you can add medicine to the mixture, which should not be hot.

Please note that all information posted on the site is for reference purposes and is not intended for independent diagnosis and treatment of diseases! Copying of materials is permitted only with an active link to the source.

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Source: http://allergiya-med.ru/preparatyi/ot-chego-lekarstvo-suprastin/

What does Suprastin help with? Instructions for use.

The drug belongs to the following groups:

Suprastin is a drug to combat allergic reactions that blocks histamine receptors. Thanks to its popularity in the pharmaceutical market, a person not even associated with medicine will now say why Suprastin is prescribed. The effect of this drug is mainly due to the suppression of the body's immune system response.

That is why doctors most often prescribe it when the question arises of how to treat allergies. Its active substance is quickly absorbed by the body and, therefore, the drug acts a short time after administration: tablets after half an hour, injections after 5-10 minutes.

What is Suprastin used for?

The main component of the drug is chloropyramine hydrochloride, which has antihistamine, sedative and antispasmodic effects. What Suprastin tablets help get rid of are allergic reactions that manifest themselves with rashes, itching, swelling, runny nose - to food, medicines, animals, insect bites. It is used during antibiotic treatment to prevent the body from reacting to the medicine.

The drug also helps with diseases accompanied by itching: hay fever, urticaria, eczema, dermatitis.

Application and contraindications

There are a number of restrictions and contraindications to the use of Suprastin. First of all, these include:

  • hypersensitivity to any of the components of the drug;
  • kidney and liver diseases (sometimes the use of the medicine is acceptable, but the dosage in such cases is reduced);
  • diseases in which taking Suprastin can cause an acute attack (for example, cardiovascular diseases, glaucoma, epilepsy);
  • respiratory failure;
  • lactose deficiency;
  • some, quite rare, metabolic disorders.

Pregnant and lactating women should not make their own decisions about taking the drug, because its action may adversely affect the health of children. It is not recommended to give Suprastin to newborns for anything - choosing a dose is very difficult, and side effects can lead to undesirable consequences. Elderly people can also take the medicine only as prescribed by a doctor - it can increase drowsiness, fatigue, and cause a drop in blood pressure.

You must be careful when using the drug. The tablets are taken with meals and washed down with water. If the doctor does not specify, the standard dosage regimen will help you navigate:

  • children aged 1 to 6 years - half a tablet 2 times a day;
  • children aged 6 to 14 years - half a tablet 2-3 times a day;
  • adults - one tablet 3-4 times a day.

Early cessation of treatment may lead to relapse of the disease. If you missed taking the pills, you should absolutely not double the dose next time - this will inevitably lead to an overdose.

If you experience symptoms such as hallucinations, loss of coordination, rapid heartbeat, or spasms, seek immediate medical attention. The patient's stomach is washed, activated charcoal is administered and the symptoms of overdose are treated. Monitoring of respiratory and cardiovascular activity is also required.

As for side effects, in addition to the usual disturbances in the functioning of the cardiovascular, digestive, and urinary systems for other drugs, Suprastin can sometimes cause:

  • a sharp and significant drop in blood pressure;
  • deterioration of blood supply to vital organs (collapse);
  • swelling of the oral cavity, difficulty breathing.

This happens with a severe overdose or individual intolerance to the drug; in such cases, hospitalization and treatment are required.

Suprastin should not be taken in parallel with drugs that act on the central nervous system, as they can enhance the effect of each other. During treatment, it is necessary to avoid alcohol, since chloropyramine is not compatible with ethanol. It is also worth temporarily limiting activities associated with risks to life and health (driving vehicles, among others), which require a person to be attentive and concentrated.

What is Suprastin used for, how and when to take it correctly - in this article we tried to cover all these issues. But still, you should consult with a therapist before starting treatment.

Look at similar drugs:

Suprastin: reviews

Before using medications, consult your doctor!

Source: http://otchegoshka.ru/suprastin-ot-chego.html

Suprastin instructions for use, analogues

The antihistamine drug Suprastin was developed more than 80 years ago. During this time, the pharmacological industry has released many new antiallergic drugs, but Suprastin is still included in the list of vital drugs.

The medicine is prescribed to adults and children, and with the appropriate dosage the drug is approved for use in the treatment of newborns.

Clinical and pharmacological group

Suprastin is an antiallergic drug related to histamine H1 receptor blockers.

Composition and release form

The main active ingredient of Suprastin is Chloropyramine hydrochloride. The drug is available in two dosage forms - in the form of tablets and in the form of a solution for injection.

Suprastin tablets are disc-shaped, white, or less often grayish in color.

One tablet contains 25 mg of active chloropyramine and additional components - gelatin, stearic acid, talc, sodium carboxymethyl starch, lactose monohydrate, potato starch.

The injection solution has a transparent color and a slight characteristic odor. One milliliter contains 20 mg of chloropyramine and water for injection.

The Suprastin solution is placed in 1 ml ampoules and is intended for intramuscular or intravenous administration.

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Pharmacological properties

Chloropyramine is a chlorinated analogue of tripelenamine, which is part of the group of ethylenediamines and belongs to the very first generation of antihistamines.

Pre-clinical and clinical trials have established the therapeutic effectiveness of chloropyramine in the treatment of patients with hay fever and a number of other allergic diseases.

Suprastin, after entering the body, blocks histamine H1 receptors. Due to this, the severity of allergy symptoms is reduced.

In addition to the antihistamine effect, Suprastin has antipruritic, hypnotic and sedative effects. The antiemetic and antispasmodic effect of taking Suprastin has been proven.

Chloropyramine affects capillary permeability, smooth muscles and central nervous system organs.

After oral administration of chloropyramine into the body, the medicine is quickly absorbed into the gastrointestinal tract. The therapeutic effect begins to develop in most patients within minutes and reaches its maximum by the end of the first hour.

The effect of Suprastin lasts from three to six hours.

Chloropyramine is metabolized by liver cells, the metabolites are excreted in the urine.

In children, Suprastin components are generally eliminated faster compared to adult patients.

The elimination of the drug is slowed down in case of impaired renal function. In patients with liver failure, the metabolism of the active substance is reduced, so they need to select the dose individually.

Indications for use

Suprastin is considered a universal antiallergic agent; its use is justified even if the specific allergen that caused the hypersensitivity reaction has not been identified.

Suprastin is included in the treatment regimen:

  • Urticaria;
  • Serum sickness;
  • Quincke's edema;
  • Seasonal and year-round forms of allergic rhinitis;
  • Allergic conjunctivitis;
  • Eczema. The drug is prescribed in both the acute and chronic stages of the disease;
  • Allergic dermatitis;
  • Allergies that develop under the influence of foods and medications;
  • Dermatitis occurring with skin itching;
  • Reactions to bites of blood-sucking insects.

Suprastin is often prescribed for the treatment of ARVI. Under its influence, the swelling of the nasal passages decreases, which makes breathing easier. The doctor determines the need to use the medicine.

Contraindications

Both tablets and the injection form of Suprastin are contraindicated:

  • With the development of an acute attack of bronchial asthma.
  • In case of hypersensitivity to one or more components of Suprastin, as well as to ethylenediamine derivatives.
  • Patients with gastric ulcer, arrhythmia, acute infarction, prostate hypertrophy, urinary retention.
  • During treatment with MAO inhibitors.
  • Women during the lactation period.

The manufacturer does not recommend prescribing Suprastin to premature infants with low body weight.

Instructions for use, dosage

The dosage of the drug, the frequency of its use and the duration of the course are determined by the doctor after examining the patient and assessing his tests.

The instructions for use contain only recommended treatment regimens for Suprastin, depending on the dosage form of the drug and the age of the patient.

Use of tablets

Suprastin tablets should be taken with meals; they should be drunk without chewing and washed down with clean water.

For adults, the daily dose of the medicine is mg, which is three to four tablets. They are drunk one at a time at regular intervals throughout the day.

For children, the dosage is:

  • From one month to one year, take ¼ tablet 2-3 times a day.
  • At the age of one to three years, the single dose is ¼ with the condition of use 3 times a day or 1/3 when taking Suprastin twice a day.
  • At the age of three to six years – a single dose of ½, take it twice a day.
  • At the ages of 6 to 14 years, the single dose is ½ Suprastin, the drug is taken 2-3 times a day.

When prescribing medication to children, it is necessary to take into account that the daily dose should not be more than 2 mg per kilogram of weight. For children, it is recommended to grind the tablet into powder and mix it with water or a small amount of regular food.

Treatment with Suprastin is stopped after the symptoms of the allergic disease have completely disappeared. The maximum dose per day for adults is 4 tablets.

The dosage of the medication is reduced or increased depending on how the person’s body responds to treatment.

Use of Suprastin in injections

Injectable Suprastin is mainly administered intramuscularly.

Intravenous injections are used once or twice to relieve severe allergic reactions and anaphylactic shock.

After intravenous injections, they move on to intramuscular use of the medication; the doctor can also replace injections with tablets.

The daily dose of Suprastin by injection is no more than 2 ml for adults.

When prescribing injections for children, their age is taken into account; the initial dose is:

  • At the age of 1 to 12 months – 0.25 ml or ¼ ampoule.
  • From one year to 6 years of age – 0.5 ml or ½ ampoule.
  • At the age of 6 to 14 years – ½ or 1 ampoule, which is 0.5 and 1 ml, respectively.

For small children, it is better to use an insulin syringe with a long needle for intramuscular administration.

If renal dysfunction is established, the dose of Suprastin is reduced. It may be less for patients with liver disease, for the elderly, and for debilitated people.

The need to reduce the dose is determined by the attending physician.

Side effects

Since Suprastin is a first-generation antihistamine, unwanted reactions may occur when taking the drug. The likelihood of their occurrence increases when the dose and frequency of medication is exceeded.

After stopping treatment, all adverse reactions disappear without the use of medications.

Most often, patients note:

  • Sedation, dizziness, fatigue, irritability, blurred vision, headache, euphoria, drowsiness. Encephalopathy, seizures, and changes in psychomotor functions may develop.
  • Arrhythmia, tachycardia, arterial hypotension.
  • Discomfort and pain in the epigastrium, dry mouth, nausea, constipation or diarrhea, changes in appetite, increased manifestations of gastroesophageal reflux. With long-term use, the development of anorexia cannot be ruled out.
  • Urinary retention and dysuria.
  • Photosensitivity.
  • Allergic reactions in the form of skin itching, urticaria, rashes. In rare cases, Quincke's edema develops.

Blood tests when taking Suprastin may show the following changes: thrombocytopenia, hemolytic anemia, leukopenia, agranulocytosis.

The likelihood of developing glaucoma and increasing intraocular pressure increases.

Overdose

Accidental or intentional overdose of Suprastin is extremely dangerous. Taking large amounts of chloropyramine can be fatal, especially for children.

  • Hallucinations;
  • Increased anxiety;
  • Impaired coordination of movements;
  • Ataxia - a violation of muscle movements;
  • Cramps.

Children with an overdose usually experience severe agitation. There is sinus tachycardia, dilated pupils, redness of the facial skin, fever, severe dry mouth, and urinary retention.

In adults, fever and hot flashes do not always occur; agitation may be accompanied by convulsions and depression.

The development of coma and cardiopulmonary collapse leads, in the absence of medical assistance, to the death of the patient within 2-18 hours.

Treatment should begin with gastric lavage. Since chloropyramine slows down the motor activity of the stomach, lavage is considered effective within 12 hours after taking a large dose of Suprastin. After this procedure, enterosorbents are prescribed.

There is no specific antidote for Suprastin, so treatment is selected based on the symptoms. Be sure to monitor the functioning of the heart and respiratory system.

Main patient groups

In pediatrics, the tablet form of the drug is most often used. In the first month of life, the drug should be used only according to indications; the need for its prescription is determined by the pediatrician.

The medicine in a minimum dosage is often prescribed from birth, excluding the period of prematurity.

For mild allergies, children are often prescribed a single dose once a day.

Suprastin is often included in the ARVI treatment regimen. The drug reduces swelling of the mucous membranes and congestion of the nasal passages.

Penetrating the blood-brain barrier, Suprastin affects the cough center, which reduces this symptom of the disease. The dosage for children is selected by the doctor.

Treatment with Suprastin for adults and children should not last more than one week. If allergy symptoms do not go away during this time, then another antihistamine is prescribed.

Suprastin is recommended for use in situations where allergies develop unexpectedly and the exact allergen is not known. With constant relapses of allergic diseases, it is necessary to use drugs that have fewer side effects.

Drug interactions

It is recommended to use Suprastin with caution simultaneously with sedatives, analgesics, tranquilizers and antidepressants, sympatholytics, and atropine.

If these medications are used with Suprastin at the same time, the likelihood of increasing their therapeutic effect increases.

Pregnancy and lactation

There have been no controlled studies on the safety of treatment with Suprastin in pregnant women. Therefore, this drug is not prescribed in the first trimester and in the last month of pregnancy.

Its use during these periods is justified only if the possible benefit of treatment with Suprastin for the mother outweighs the likely risk of negative effects on the fetus.

If there is a need to use the drug during the lactation period, then breastfeeding should be suspended for the period of therapy.

special instructions

The instructions for use of Suprastin indicate that this antihistamine, when used simultaneously with ototoxic drugs, can mask the first signs indicating a hearing impairment.

Taking the drug in the evening sometimes increases the manifestations of reflux esophagitis. Therefore, patients with this disease should take the medicine several hours before bedtime.

Suprastin has the ability to enhance the effect of ethanol on the central nervous system. In this regard, when treating with this drug, alcohol intake should be completely avoided.

Each Suprastin tablet contains 116 mg of lactose monohydrate. This amount is sufficient to cause undesirable changes in well-being in people with lactase deficiency, galactosemia, and galactose/glucose malabsorption syndrome.

Suprastin often leads to increased fatigue, dizziness and drowsiness. These reactions are especially pronounced at the initial stage of treatment.

In this regard, patients are prohibited from working on complex mechanisms or driving vehicles in the first days of therapy. In the future, these restrictions may be lifted, but this is decided only by the doctor.

For liver and kidney dysfunction

If there are pathologies of the liver and kidneys, the patient must notify the attending physician in advance. Depending on the degree of dysfunction of these organs, it may be necessary to select an individual dose; most often, the dosage of Suprastin is reduced.

The likelihood of developing severe drowsiness and dizziness is increased in older people and in malnourished people. Therefore, Suprastin is prescribed to these categories of patients with caution or replaced with a safer analogue.

Conditions of storage and dispensing in pharmacies

Both the tablets and the ampoule should be stored in places protected from light at a temperature of no more than 25 degrees.

Suprastin ampoules should be sold in pharmacies upon presentation of a prescription from a doctor. The tablets are also approved for over-the-counter release.

Analogs

Analogs of Suprastin based on the active substance include drugs such as:

According to the mechanism of action, the main analogues of Suprastin are Diphenhydramine, Tavegil, Diazolin, Claritin, Cetrin, Zyrtek.

Reviews

“Suprastin has become a permanent drug in our home medicine cabinet since it turned out that our youngest son is allergic. Moreover, he could react with rapidly increasing swelling of the lips and eyes, sometimes to no one knows why.

The first time we were so afraid that the ambulance wouldn’t make it in time, as our son began to fall asleep right in our arms. The doctor arrived and quickly gave several injections, including Suprastin.

After the examination, we were prescribed treatment, and the allergist advised us to buy Suprastin in tablets and keep it on hand at all times.

If an allergic reaction occurs, I immediately give my son half of the tablet, after crushing it into powder and diluting it with juice.

Allergy symptoms begin to decrease within just half an hour. A few hours later I give him a second rug and after that I’m not afraid that Quincke’s edema will occur.

Naturally, Suprastin has many disadvantages, but this is the only drug that suited us as a first aid remedy.

We don’t use it for a long time - the maximum treatment lasts 5 days, then, if necessary, we switch to other antihistamines.”

“That summer, I was bitten in the area near my eye by some kind of insect. At first I didn’t attach any importance to it, I thought it would scratch and go away. But by the evening my eye was almost completely swollen, the swelling began to go down, and severe lacrimation appeared.

My neighbor at the dacha gave me Suprastin and told me to take a whole pill at once, which I did. After about two hours, it became noticeable that the eye was opening and I was no longer so afraid to fall asleep.”

“For the fourth year in a row, at the beginning of summer I have had allergic rhinitis, which I haven’t identified specifically yet.

Nasal congestion, runny nose, and paroxysmal sneezing continue for two to three weeks, then gradually disappear.

During those years, I received practically no treatment, since I was pregnant then and then breastfed the child.

This summer I decided not to suffer from discomfort and began treatment with Suprastin almost immediately after the onset of a runny nose.

The drug helped, after taking the second tablet there was only a small discharge left.

But on the second day of treatment, I began to suffer from severe drowsiness and fatigue, and in the evening I developed a headache.

These adverse reactions were even worse than the allergy itself, so Suprastin had to be abandoned. I hope that in the spring I will still find time to visit an allergist so that he can prescribe me the appropriate medications.”

Maria Ivanovna, 52 years old.

“Suprastin always helps me if food allergies occur. The drug not only eliminates nausea, itching in the mouth and colic, but also relieves skin rashes and itching on the body. All manifestations decrease within an hour after the tablet is taken.

Disadvantages include a bitter, astringent taste and the need to take the medicine 3-4 times a day.”

“My husband and I, like our children, are not prone to allergic reactions. But as they say, there’s nothing you can’t deny.

It so happened that our eldest daughter had not consumed any products with cinnamon since birth and therefore we could not think that she would be allergic to this seasoning.

After eating cinnamon rolls, a few hours later our girl began to cry, complain of stomach pain, she even vomited, and by the evening a rash appeared on her body.

We went to the children's hospital ourselves, the doctor examined us and immediately said that it was a food allergy. Right there they gave me Suprastin as an injection and prescribed me to drink activated charcoal.

After the injection, my daughter calmed down almost immediately, and when she arrived home she fell asleep soundly.

We drank Suprastin tablets and activated charcoal for three days, during which time all the symptoms of the reaction disappeared. Now we always have this medicine in our medicine cabinet, but there is no cinnamon in the house.”

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